Attribute | Details |
---|---|
Generic Name | Bicalutamide |
Dosage Forms | 50mg tablets |
Pharmacological Class | Antiandrogen |
Primary Use | Prostate cancer treatment |
Mechanism of Action | Blocks androgen receptors |
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Chemical Structure
The chemical compound bicalutamide underlies Casodex 50mg. It falls into the class of non-steroidal antiandrogens. The structure of bicalutamide comprises a racemic mixture. One enantiomer holds therapeutic relevance. The other remains largely inactive.
Bicalutamide’s molecular formula is C18H14F4N2O4S. Its configuration contains trifluoromethyl groups and a thioester linkage. This architecture aids in receptor binding, crucial for its mode of action. The presence of fluorine atoms enhances metabolic stability.
Casodex’s design allows it to bind with androgen receptors. This property hinders androgen-driven tumor growth. Its selective affinity mitigates adverse impacts on other steroid receptors.
Casodex Use
Casodex 50mg addresses advanced prostate cancer. It is frequently combined with other therapies, including luteinizing hormone-releasing hormone analogs. The goal remains halting disease progression.
Patients with metastatic prostate cancer benefit from Casodex. It serves as a vital part of androgen deprivation therapy. The pharmaceutical effectively competes with natural hormones. This competition reduces cancer cell proliferation.
Prescription relies on thorough evaluation by healthcare professionals. A patient’s overall health status is critical for determining suitability.
Casodex Contraindications
Casodex is contraindicated in several conditions. Women and children must avoid this medication. Patients with known hypersensitivity to bicalutamide are also at risk.
Individuals with severe liver impairment should not use Casodex 50mg. The liver metabolizes the drug significantly. Compromised hepatic function increases toxicity risks.
Concomitant use with terfenadine, astemizole, or cisapride is inadvisable. Such combinations potentially induce severe cardiac events. Precautions are necessary for patients with cardiac history.
Casodex Disposal
Proper disposal of Casodex is vital to ensure safety. Unused or expired tablets should not enter household trash or water systems. Doing so could harm the environment or others.
Return unused medications to pharmacies offering take-back services. Some communities hold drug take-back events for proper disposal.
Patients must follow local guidelines for disposal. For further guidance, consult a pharmacist or local waste management authorities.
Casodex Side Effects
Casodex 50mg may cause various side effects. Common issues include hot flashes, nausea, and breast tenderness. These symptoms often resolve with continued therapy.
Serious adverse effects demand immediate medical attention. Liver function alterations, jaundice, and severe abdominal pain are critical. Prompt intervention can prevent complications.
Monitoring blood counts during therapy is advisable. Patients should report any unusual bruising or bleeding to their physician.
Casodex Over The Counter
Casodex is not available over the counter. It requires a prescription from a healthcare professional. This restriction ensures patient safety and efficacy of treatment.
Patients should not seek alternative or online sources without consulting their doctor. Unauthorized suppliers might offer counterfeit products, risking health.
Comprehensive care includes ongoing consultations and regular assessments. Professional guidance optimizes treatment outcomes and minimizes risks.